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 FDA - Approved

 

HIV and AIDS Treatments
October 24, 2006

 

Source:  www.HIVandHepatitis.com

 

Protease Inhibitors
Agenerase (amprenavir)
Aptivus (tipranavir)
Crixivan (indinavir)
Fortovase (saquinavir soft gel)
Invirase (saquinavir hard gel)
Kaletra (lopinavir/ritronavir)
Lexiva (Fosamprenavir)
Norvir (ritonavir)
Prezista (darunavir)
Reyataz (atazanavir)
Viracept (nelfinavir)

Nucleoside / Nucleotide Reverse Transcriptase Inhibitors

Combivir (AZT 3TC)
Epivir (lamivudine; 3TC)
Emtriva (emtricitabine; FTC)
Epzicom (abacavir lamivudine)
Hivid (zalcitabine; ddC)
Retrovir (zidovudine; AZT)
Trizivir (abacavir zidovudine lamivudine)
Truvada  (Tenofovir / Emtricitabine)
Videx (didanosine; ddI)
Viread (tenofovir)

Zerit (stavudine; d4T)
Ziagen (abacavir)


non Nucleoside Reverse Transcriptase Inhibitors
Rescriptor (delavirdine)

Sustiva (efavirenz)
Viramune (nevirapine)

Entry Inhibitors
Fuzeon (enfuvirtide; T-20)

Fixed-dose Combinations
Atripla
(efavirenz emtricitabine tenofovir)
Combivir
(retrovir lamivudine)

Trizivir
(abacavir zidovudine lamivudine)
Truvada
(tenofovir emtricitabine)

FDA-approved Anti-HIV Drugs
 
 Protease Inhibitors (PI)
 Non Nucleoside Reverse Transcriptase Inhibitors (nNRTI)
 Nucleoside/Nucleotide Reverse Transcriptase Inhibitors (NRTI)
 Entry / Fusion Inhibitors (EI)
 Fixed-dose Combinations
 New Fact Sheet Lists Formulations Available for All FDA-approved Anti-HIV Drugs
 Experimental Treatments Chart
Sponsors
 

Nucleoside / Nucleotide
Reverse Transcriptase
Inhibitors

 


Protease Inhibitors

 


non Nucleoside Reverse Transcriptase Inhibitors


Entry Inhibitors
Combivir
(AZT plus 3TC)

Epivir
(lamivudine; 3TC)

Emtriva
(emtricitabine; FTC)

Hivid
(zalcitabine; ddC)

Retrovir
(zidovudine; AZT)

Trizivir
(abacavir plus zidovudine plus lamivudine)


Truvada
(Tenofovir Emtricitabine)


Videx
(didanosine; ddI)

Viread
(tenofovir)


Zerit
(stavudine; d4T)

Ziagen
(abacavir)

 

Agenerase
(amprenavir)

Aptivus
(tipranavir)

Crixivan
(indinavir)

Fortovase
(saquinavir soft gel capsules)

Invirase
(saquinavir hard gel capsules)


Kaletra
(lopinavir/ritronavir)



Lexiva

(Fosamprenavir)

Norvir
(ritonavir)


Prezista
(darunavir)


Reyataz
(atazanavir)

Viracept
(nelfinavir)

Rescriptor
(delavirdine)


Sustiva
(efavirenz)

Viramune
(nevirapine)
Fuzeon
(enfuvirtide; T-20)

 

Fixed-dose Combinations

 

Atripla
(efavirenz emtricitabine tenofovir)

Combivir
(retrovir lamivudine)


Epzicom
(abacavir lamivudine)

Trizivir
(abacavir zidovudine lamivudine)

Truvada
(tenofovir emtricitabine)

 

 

 

 

 

 

 




 

 

 

 

 
Protease Inhibitors  (PI) TOP  
Brand Name
Generic Names
Abbreviation
Manufacturer
amprenavir
APV
GlaxoSmithKline
  Aptivus Tipranavir TPV Boehringer Ingelheim
indinavir
IDV
Merck
saquinavir (soft gel cap)
SQV (SGC)
Roche
saquinavir (hard gel cap)
SQV (HGC)
Roche
  Kaletra
lopinavir/ritonavir
LPV/r
Abbott Laboratories
  Lexiva
fosamprenavir
FPV
GlaxoSmithKline
  Norvir
ritonavir
RTV
Abbott Laboratories
  Prezista
darunavir   Tibotec
  Reyataz
atazanavir
ATV
Bristol-Myers Squibb
nelfinavir
NFV
Pfizer

 

  Ritonavir-boosted Protease Inhibitors
  
Guide to Management of Toxicities and Side Effects of Protease Inhibitors [PDF]

 

 

 Non Nucleoside Reverse Transcriptase Inhibitors (nNRTI) TOP  
Brand Name
Generic Names
Abbreviation
Manufacturer
  Rescriptor delavirdine
DLV
Pfizer
  Sustiva efavirenz
EFV
Bristol-Myers Squibb
  Viramune nevirapine
NVP
Boehringer Ingelheim

 

  Guide to Management of Toxicities and Side Effects of nNRTIs [PDF]

 

 

 Nucleoside / Nucleotide Reverse Transcriptase Inhibitors  (NRTI) TOP  
Brand Name
Generic Names
Abbreviation
Manufacturer
  Combivir zidovudine lamivudine
AZT 3TC
GlaxoSmithKline
  Emtriva emtricitabine
FTC
Gilead Sciences
  Epivir lamivudine
3TC
GlaxoSmithKline
  Epzicom abacavir lamivudine
ABC 3TC
GlaxoSmithKline
  Hivid zalcitabine
ddC
Roche
  Retrovir zidovudine
AZT or ZDV
GlaxoSmithKline
  Trizivir abacavir zidovudine lamivudine
ABC AZT 3TC
GlaxoSmithKline
  Truvada tenofovir emtricitabine
TDF FTC
Gilead Sciences
  VIDEX didanosine
ddI
Bristol-Myers Squibb
  VIDEX EC didanosine: delayed-release capsules
ddI
Bristol-Myers Squibb
  Viread tenofovir DF TDF Gilead Sciences
  Zerit stavudine
d4T
Bristol-Myers Squibb
  Zerit XR stavudine: delayed-release
d4T
Bristol-Myers Squibb
  Ziagen abacavir
ABC
GlaxoSmithKline

 

  Guide to Management of Toxicities and Side Effects of NRTIs [PDF}

 

 

 Entry / Fusion Inhibitors TOP  
Brand Name
Generic Names
Abbreviation
Manufacturer
  Fuzeon enfuvirtide
ENF
Roche / Trimeris
 
 Fixed-dose Combinations TOP  
Brand Name
Generic Names
Abbreviation
Manufacturer
  Atripla
efavirenz emtricitabine tenofovir EFV FTC TDF Gilead Sciences
Bristol-Myers Squibb
  Combivir zidovudine lamivudine AZT 3TC GlaxoSmithKline
  Epzicom abacavir lamivudine ABC 3TC GlaxoSmithKline
  Trizivir abacavir zidovudine lamivudine ABC AZT 3TC GlaxoSmithKline
  Truvada tenofovir emtricitabine TDF FTC Gilead Sciences